Access to High Levels of Molecular Complexity by One-Pot Iridium/Enamine Asymmetric Catalysis

Independent workers with team spirit: A catalytic sequence that exploits the compatibility of (chiral) cationic iridium catalysts for the isomerization of primary allylic alcohols to aldehydes with organocatalysts has been developed for the highly enantioselective alpha functionalization of aldehydes (up to 66 % yield, d.r. 49:1, 99 % ee). The reaction displayed useful generality with respect to both the nucleophile and the electrophile.

Références

Titre
Access to High Levels of Molecular Complexity by One-Pot Iridium/Enamine Asymmetric Catalysis
Type de publication
Article de revue
Année de publication
2011
Revue
Angewandte Chemie International Edition
Volume
50
Ticket
10
Pagination
2354–2358
Soumis le 7 septembre 2022