Département de chimie moléculaire

Chemobacterial Synthesis of a Sialyl-Tn Cyclopeptide Vaccine Candidate., Richard, Emeline, Pifferi Carlo, Fiore Michele, Samain Eric, Le Gouellec Audrey, Fort Sebastien, Renaudet Olivier, and Priem Bernard. , ChemBioChem, Volume 18, Number 17, p.1730–1734, (2017)

Cyclopeptide scaffolds in carbohydrate-based synthetic vaccines., Pifferi, Carlo, Berthet Nathalie, and Renaudet Olivier , Biomater. Sci., Volume 5, Number 5, p.953–965, (2017)

Heterovalent Glycodendrimers as Epitope Carriers for Antitumor Synthetic Vaccines., Pifferi, Carlo, Thomas Baptiste, Goyard David, Berthet Nathalie, and Renaudet Olivier , Chem. - A Eur. J., Volume 23, Number 64, p.16283–16296, (2017)

Immunological characterization of a rigid $\alpha$-Tn mimetic on murine iNKT and human NK cells., Fallarini, Silvia, Brittoli Alvaro, Fiore Michele, Lombardi Grazia, Renaudet Olivier, Richichi Barbara, and Nativi Cristina. , Glycoconj. J., Volume 34, Number 4, p.553–562, (2017)

An oxime-based glycocluster microarray., Hoang, Antoine, Laigre Eugenie, Goyard David, Defrancq Eric, Vinet Francoise, Dumy Pascal, and Renaudet Olivier , Org. Biomol. Chem., Volume 15, Number 24, p.5135–5139, (2017)

Synthesis of Mannosylated Glycodendrimers and Evaluation against BC2L-A Lectin from Burkholderia Cenocepacia., Pifferi, Carlo, Goyard David, Gillon Emilie, Imberty Anne, and Renaudet Olivier , Chempluschem, Volume 82, Number 3, p.390–398, (2017)

Identification of Nanomolar Lectin Ligands by a Glycodendrimer Microarray., Laigre, Eugenie, Tiertant Claire, Goyard David, and Renaudet Olivier , ACS Omega, Volume 3, Number 10, p.14013–14020, (2018)

Multivalent Glycomimetics with Affinity and Selectivity toward Fucose-Binding Receptors from Emerging Pathogens., Goyard, David, Baldoneschi Veronica, Varrot Annabelle, Fiore Michele, Imberty Anne, Richichi Barbara, Renaudet Olivier, and Nativi Cristina. , Bioconjug. Chem., Volume 29, Number 1, p.83–88, (2018)

The study of multivalent carbohydrate-protein interactions by bio-layer interferometry., Laigre, Eugenie, Goyard David, Tiertant Claire, Dejeu Jérôme, and Renaudet Olivier , Org. Biomol. Chem., Volume 16, Number 46, p.8899–8903, (2018)

Tailor-made Janus lectin with dual avidity assembles glycoconjugate multilayers and crosslinks protocells., Ribeiro, Joao P., Villringer Sarah, Goyard David, Guerente Liliane, Hoferlin Manuela, Renaudet Olivier, Romer Winfried, and Imberty Anne. , Chem. Sci., Volume 9, Number 39, p.7634–7641, (2018)

Heteroglycoclusters With Dual Nanomolar Affinities for the Lectins LecA and LecB From Pseudomonas aeruginosa, Goyard, David, Thomas Baptiste, Gillon Emilie, Imberty Anne, and Renaudet Olivier , Frontiers in Chemistry, Volume 7, p.666, (2019)

Multifunctional Glycoconjugates for Recruiting Natural Antibodies against Cancer Cells, Liet, Benjamin, Laigre Eugenie, Goyard David, Todaro Biagio, Tiertant Claire, Boturyn Didier, Berthet Nathalie, and Renaudet Olivier , Chemistry – A European Journal, Volume 25, p.15508-15515, (2019)

Multifunctional Glycoconjugates for Recruiting Natural Antibodies against Cancer Cells., Liet, Benjamin, Laigre Eugenie, Goyard David, Todaro Biagio, Tiertant Claire, Boturyn Didier, Berthet Nathalie, and Renaudet Olivier , Chem. - Eur. J., Volume 25, p.15508–15515, (2019)

Multivalent glycoligands with lectin/enzyme dual specificity: self-deliverable glycosidase regulators., Gonzalez-Cuesta, Manuel, Goyard David, Nanba Eiji, Higaki Katsumi, Fernandez Jose M. Garcia, Renaudet Olivier, and Mellet Carmen. Ortiz , Chem. Commun. (Cambridge, U. K.), Volume 55, p.12845–12848, (2019)

Multivalent glycoligands with lectin/enzyme dual specificity: self-deliverable glycosidase regulators, Gonzalez-Cuesta, Manuel, Goyard David, Nanba Eiji, Higaki Katsumi, Fernandez Jose M. Garcia, Renaudet Olivier, and Mellet Carmen Ortiz , Chem. Commun., Volume 55, p.12845-12848, (2019)

Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2, Roussel, Emile, Tran-Nguyen Viet-Khoa, Bouhedjar Khalid, Dems Mohamed Abdesselem, Belaidi Amine, Matougui Brahim, Peres Basile, Azioune Ammar, Renaudet Olivier, Falson Pierre, et al. , European Journal of Medicinal Chemistry, Volume 184, p.111772, (2019)

Optimization of the chromone scaffold through QSAR and docking studies: identification of potent inhibitors of ABCG2., Roussel, Emile, Tran-Nguyen Viet-Khoa, Bouhedjar Khalid, Dems Mohamed Abdesselem, Belaidi Amine, Matougui Brahim, Peres Basile, Azioune Ammar, Renaudet Olivier, Falson Pierre, et al. , Eur. J. Med. Chem., Volume 184, p.111772, (2019)

Selective high-resolution DNP-enhanced NMR of biomolecular binding sites, Marin-Montesinos, Ildefonso, Goyard David, Gillon Emilie, Renaudet Olivier, Imberty Anne, Hediger Sabine, and De Paepe Gael , Chem. Sci., Volume 10, p.3366-3374, (2019)

Towards the preparation of synthetic outer membrane vesicle models with micromolar affinity to wheat germ agglutinin using a dialkyl thioglycoside, Fayolle, Dimitri, Berthet Nathalie, Doumeche Bastien, Renaudet Olivier, Strazewski Peter, and Fiore Michele , Beilstein Journal of Organic Chemistry, Volume 15, p.937-946, (2019)

Towards the preparation of synthetic outer membrane vesicle models with micromolar affinity to wheat germ agglutinin using a dialkyl thioglycoside., Fayolle, Dimitri, Berthet Nathalie, Doumeche Bastien, Renaudet Olivier, Strazewski Peter, and Fiore Michele. , Beilstein J. Org. Chem., Volume 15, p.937–946, (2019)

Chemical synthesis and immunological evaluation of new generation multivalent anticancer vaccines based on a Tn antigen analogue, Pifferi, Carlo, Ruiz-de-Angulo Ane, Goyard David, Tiertant Claire, Sacristán Nagore, Barriales Diego, Berthet Nathalie, Anguita Juan, Renaudet Olivier, and Fernández-Tejada Alberto , Chem. Sci., 04/2020, Volume 11, p.4488 - 4498 , (2020)

Development of C-type lectin-oriented surfaces for high avidity glycoconjugates: towards mimicking multivalent interactions on the cell surface, Porkolab, Vanessa, Pifferi Carlo, Sutkeviciute Ieva, Ordanini Stefania, Taouai Marwa, Thepaut Michel, Vivès Corinne, Benazza Mohammed, Bernardi Anna, Renaudet Olivier, et al. , Org. Biomol. Chem., 06/2020, Volume 18, p.4763 - 4772, (2020)

Antibody recruiting molecules (ARMs): synthetic immunotherapeutics to fight cancer, Achilli, Silvia, Berthet Nathalie, and Renaudet Olivier , RSC Chem. Biol., 03/2021, Volume 2, p.713-724 , (2021)

Clicked Bifunctional Dendrimeric and Cyclopeptidic Addressable Redox Scaffolds for the Functionalization of Carbon Nanotubes with Redox Molecules and Enzymes, Gentil, S., Pifferi C., Rousselot-Pailley P., Tron T., Renaudet Olivier, and Le Goff Alan , Langmuir, Volume 37, Issue 3, (2021)

Clicked Bifunctional Dendrimeric and Cyclopeptidic Addressable Redox Scaffolds for the Functionalization of Carbon Nanotubes with Redox Molecules and Enzymes, Gentil, Solène, Pifferi Carlo, Rousselot-Pailley Pierre, Tron Thierry, Renaudet Olivier, and Le Goff Alan , Langmuir, 01/2021, Volume 37, p.1001-1011, (2021)

Multivalent Presentations of Glycomimetic Inhibitor of the Adhesion of Fungal Pathogen Candida albicans to Human Buccal Epithelial Cells, Martin, Harlei, Goyard David, Margalit Anatte, Doherty Kyle, Renaudet Olivier, Kavanagh Kevin, and Velasco-Torrijos Trinidad , Bioconjugate Chemistry, 04/2021, Volume 32, Issue 5, p.971–982, (2021)

Structural influence of antibody recruiting glycodendrimers (ARGs) on antitumoral cytotoxicity, Todaro, Biagio, Achilli Silvia, Liet Benjamin, Laigre Eugenie, Tiertant Claire, Goyard David, Berthet Nathalie, and Renaudet Olivier , Biomater. Sci., 04/2021, Volume 9, p.4076-4085 , (2021)

Characterization of the interaction of multivalent glycosylated ligands with bacterial lectins by BioLayer interferometry, Picault, L, Laigre E, Gillon E, Tiertant C, Renaudet Olivier, Imberty A, Goyard David, and Dejeu J , Glycobiology, 07/2022, Volume 32, Issue 10, p.886-896, (2022)

Cyclopeptides as glycan-presenting multivalent scaffolds, Goyard, David, and Renaudet Olivier , Carbohydrate Chemistry: Chemical and Biological Approaches, Volume 45, p.499-518, (2022)

Homo- and Heterovalent Neoglycoproteins as Ligands for Bacterial Lectins, Goyard, David, Roubinet Benoît, Vena Federica, Landemarre Ludovic, and Renaudet Olivier , ChemPlusChem, Volume 87, p.e202100481, (2022)

Multivalent glycocyclopeptides: conjugation methods and biological applications, Goyard, David, Martin-Serrano-Ortiz Angela, Boturyn Didier, and Renaudet Olivier , Chem. Soc. Rev., 10/2022, Volume 51, p.8756 – 8783, (2022)

Targeting Tn-Antigen-Positive Human Tumors with a Recombinant Human Macrophage Galactose C-Type Lectin, Bulteau, François, Thepaut Michel, Henry Maxime, Hurbin Amandine, Vanwonterghem Laetitia, Vivès Corinne, Le Roy Aline, Ebel Christine, Renaudet Olivier, Fieschi Franck, et al. , Molecular Pharmaceutics, Volume 19, p.235-245, (2022)

Advanced high-affinity glycoconjugate ligands of galectins, Hovorková, Michaela, Červený Jakub, Bumba Ladislav, Pelantová Helena, Cvačka Josef, Křen Vladimír, Renaudet Olivier, Goyard David, and Bojarová Pavla , Bioorganic Chemistry, 11/2022, Volume 131, p.106279, (2023)