Département de chimie moléculaire

Novel synthetic bis-indolic derivatives with antistaphylococcal activity, including against MRSA and VISA strains., Caspar, Yvan, Jeanty Matthieu, Blu Jérôme, Burchak Olga, Le Pihive Emmanuelle, Maigre Laure, Schneider Dominique, Jolivalt Claude, Paris Jean-Marc, Hequet Arnaud, et al. , J. Antimicrob. Chemother., Volume 70, Number 6, p.1727–1737, (2015)

1-(1H-Indol-3-yl)ethanamine Derivatives as Potent Staphylococcus aureus NorA Efflux Pump Inhibitors., Hequet, Arnaud, Burchak Olga N., Jeanty Matthieu, Guinchard Xavier, Le Pihive Emmanuelle, Maigre Laure, Bouhours Pascale, Schneider Dominique, Maurin Max, Paris Jean-Marc, et al. , ChemMedChem, Volume 9, Number 7, p.1534–1545, (2014)

Bis-indolic compounds as potential new therapeutic alternatives for tularaemia., Caspar, Yvan, Sutera Vivien, Boisset Sandrine, Denis Jean-Noël, and Maurin Max. , Front. Cell. Infect. Microbiol., Volume 4, p.24/1–24/7, (2014)

Concise preparation of optically active heteroaryl α-(hydroxyamino) esters., Murat-Onana, Marie Laure, Berini Christophe, Denis Jean-Noël, Poisson Jean-François, Minassian Frédéric, and Pelloux-Leon Nadia , Eur. J. Org. Chem., Volume 2014, Number 18, p.3773–3776, (2014)

Synthesis and evaluation of 1-(1H-indol-3-yl)ethanamine derivatives as new antibacterial agents., Burchak, Olga N., Le Pihive Emmanuelle, Maigre Laure, Guinchard Xavier, Bouhours Pascale, Jolivalt Claude, Schneider Dominique, Maurin Max, Giglione Carmela, Meinnel Thierry, et al. , Bioorg. Med. Chem., Volume 19, Number 10, p.3204–3215, (2011)

An efficient method for the synthesis of unsymmetrical 2,2'-bis(pyrrolyl)alkanes., Murat-Onana, Marie Laure, Berini Christophe, Minassian Frédéric, Pelloux-Leon Nadia, and Denis Jean-Noël , Org. Biomol. Chem., Volume 8, Number 9, p.2204–2211, (2010)

From N-triisopropylsilylpyrrole to an optically active C-4 substituted pyroglutamic acid: total synthesis of penmacric acid., Berini, Christophe, Pelloux-Leon Nadia, Minassian Frédéric, and Denis Jean-Noël , Org. Biomol. Chem., Volume 7, Number 21, p.4512–4516, (2009)

Efficient stereoselective nucleophilic addition of pyrroles to chiral nitrones., Berini, Christophe, Minassian Frédéric, Pelloux-Leon Nadia, Denis Jean-Noël, Vallee Yannick., and Philouze Christian , Org. Biomol. Chem., Volume 6, Number 14, p.2574–2586, (2008)

Expanding the chemical diversity of CK2 inhibitors., Prudent, Renaud, Moucadel Virginie, Lopez-Ramos Miriam, Aci Samia, Laudet Beatrice, Mouawad Liliane, Barette Caroline, Einhorn Jacques, Einhorn Cathy, Denis Jean-Noël, et al. , Mol. Cell. Biochem., Volume 316, Number 1{&}2, p.71–85, (2008)

Heterolignans: Stereoselective synthesis of an 11-amino analog of azaelliptitoxin., Routier, Julie, Calancea Mihaela, David Marion, Vallee Yannick., and Denis Jean-Noël , European J. Org. Chem., Number 34, p.5687–5691, (2008)

Reactions of In Situ Generated N-Boc Nitrones with Aromatic and Heteroaromatic Grignard Reagents: Application to the Synthesis of Zileuton., Guinchard, Xavier, and Denis Jean-Noël , J. Org. Chem., Volume 73, Number 5, p.2028–2031, (2008)

Total Syntheses of Brominated Marine Sponge Alkaloids., Guinchard, Xavier, Vallee Yannick., and Denis Jean-Noël , Org. Lett., Volume 9, Number 19, p.3761–3764, (2007)

Total Synthesis of Marine Sponge Bis(indole) Alkaloids of the Topsentin Class., Guinchard, Xavier, Vallee Yannick., and Denis Jean-Noël , J. Org. Chem., Volume 72, Number 10, p.3972–3975, (2007)