Département de chimie moléculaire

Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2, Roussel, Emile, Tran-Nguyen Viet-Khoa, Bouhedjar Khalid, Dems Mohamed Abdesselem, Belaidi Amine, Matougui Brahim, Peres Basile, Azioune Ammar, Renaudet Olivier, Falson Pierre, et al. , European Journal of Medicinal Chemistry, Volume 184, p.111772, (2019)

Optimization of the chromone scaffold through QSAR and docking studies: identification of potent inhibitors of ABCG2., Roussel, Emile, Tran-Nguyen Viet-Khoa, Bouhedjar Khalid, Dems Mohamed Abdesselem, Belaidi Amine, Matougui Brahim, Peres Basile, Azioune Ammar, Renaudet Olivier, Falson Pierre, et al. , Eur. J. Med. Chem., Volume 184, p.111772, (2019)

Orthogonal dual thiol-chloroacetyl and thiol-ene coupling for the sequential one-pot assembly of heteroglycoclusters., Fiore, Michele, Daskhan Gour Chand, Thomas Baptiste, and Renaudet Olivier , Beilstein J. Org. Chem., Volume 10, p.1557–1563, 7 pp., (2014)

Oxime Ligation: A Chemoselective Click-Type Reaction for Accessing Multifunctional Biomolecular Constructs., Ulrich, Sebastien, Boturyn Didier, Marra Alberto, Renaudet Olivier, and Dumy Pascal , Chem. - A Eur. J., Volume 20, Number 1, p.34–41, (2014)

An oxime-based glycocluster microarray., Hoang, Antoine, Laigre Eugenie, Goyard David, Defrancq Eric, Vinet Francoise, Dumy Pascal, and Renaudet Olivier , Org. Biomol. Chem., Volume 15, Number 24, p.5135–5139, (2017)

Oxime-based synthesis of new chromogenic and fluorogenic oligosaccharides., Renaudet, Olivier, and Dumy Pascal , European J. Org. Chem., Number 32, p.5383–5386, (2008)

Phenolic oxime oligomers inhibit Alzheimer's amyloid fibril formation and disaggregate fibrils in vitro., Dolphin, Gunnar T., Renaudet Olivier, Ouberai Myriam, Dumy Pascal, Garcia Julian, and Reymond Jean-Louis. , ChemBioChem, Volume 10, Number 8, p.1325–1329, (2009)

Promotion of sugar-lectin recognition through the multiple sugar presentation offered by regioselectively addressable functionalized templates (RAFT): a QCM-D and SPR study., Wilczewski, Marie, Van der Heyden Angeline, Renaudet Olivier, Dumy Pascal, Guerente Liliane, and Labbe Pierre , Org. Biomol. Chem., Volume 6, Number 6, p.1114–1122, (2008)

RAFT Nano-constructs: surfing to biological applications., Boturyn, Didier, Defrancq Eric, Dolphin Gunnar T., Garcia Julian, Labbe Pierre, Renaudet Olivier, and Dumy Pascal , J. Pept. Sci., Volume 14, Number 2, p.224–240, (2008)

Randomized Combinatorial Library of Hetero-glyco-clusters (hGC)., Dulery, Vincent, Renaudet Olivier, Wilczewski Marie, Van der Heyden Angeline, Labbe Pierre, and Dumy Pascal , J. Comb. Chem., Volume 10, Number 3, p.368–371, (2008)

Recent advances on cyclopeptide-based glycoclusters., Renaudet, Olivier , Mini. Rev. Org. Chem., Volume 5, Number 4, p.274–286, (2008)

Re-evaluation of binding properties of recombinant lymphocyte receptors NKR-P1A and CD69 to chemically synthesized glycans and peptides., Rozbesky, Daniel, Krejzova Jana, Krenek Karel, Prchal Jan, Hrabal Richard, Kozisek Milan, Weignerova Lenka, Fiore Michele, Dumy Pascal, Renaudet Olivier, et al. , Int. J. Mol. Sci., Volume 15, Number 1, p.1271–1283, 13 pp., (2014)

Role of a Preorganized Scaffold Presenting Four Residues of a GM-3 Lactone Mimetic on Melanoma Progression., Richichi, Barbara, Comito Giuseppina, Renaudet Olivier, Fiore Michele, Marra A, Stecca B, Pasquato L, Chiarugi P, and Nativi C , ACS Med. Chem. Lett., Volume 7, Number 1, p.28–33, (2016)

Selective high-resolution DNP-enhanced NMR of biomolecular binding sites, Marin-Montesinos, Ildefonso, Goyard David, Gillon Emilie, Renaudet Olivier, Imberty Anne, Hediger Sabine, and De Paepe Gael , Chem. Sci., Volume 10, p.3366-3374, (2019)

Structural influence of antibody recruiting glycodendrimers (ARGs) on antitumoral cytotoxicity, Todaro, Biagio, Achilli Silvia, Liet Benjamin, Laigre Eugenie, Tiertant Claire, Goyard David, Berthet Nathalie, and Renaudet Olivier , Biomater. Sci., 04/2021, Volume 9, p.4076-4085 , (2021)

Structure-based design of small peptide inhibitors of protein kinase CK2 subunit interaction., Laudet, Beatrice, Barette Caroline, Dulery Vincent, Renaudet Olivier, Dumy Pascal, Metz Alexandra, Prudent Renaud, Deshiere Alexandre, Dideberg Otto, Filhol Odile, et al. , Biochem. J., Volume 408, Number 3, p.363–373, (2007)

The study of multivalent carbohydrate-protein interactions by bio-layer interferometry., Laigre, Eugenie, Goyard David, Tiertant Claire, Dejeu Jérôme, and Renaudet Olivier , Org. Biomol. Chem., Volume 16, Number 46, p.8899–8903, (2018)

Surface patterning of (bio)molecules onto the inner wall of fused-silica capillary tubes., Dendane, Nabil, Hoang Antoine, Renaudet Olivier, Vinet Francoise, Dumy Pascal, and Defrancq Eric , Lab Chip, Volume 8, Number 12, p.2161–2163, (2008)

Synthesis of a New Series of Sialylated Homo- and Heterovalent Glycoclusters by using Orthogonal Ligations., Daskhan, Gour Chand, Pifferi Carlo, and Renaudet Olivier , ChemistryOpen, Volume 5, Number 5, p.477–484, (2016)

Synthesis of Glycocyclopeptides by Click Chemistry and Inhibition Assays with Lectins., Bossu, Isabelle, Berthet Nathalie, Dumy Pascal, and Renaudet Olivier , J. Carbohydr. Chem., Volume 30, Number 7-9, p.458–468, (2011)

Synthesis of heteroglycoclusters by using orthogonal chemoselective ligations., Thomas, Baptiste, Fiore Michele, Bossu Isabelle, Dumy Pascal, and Renaudet Olivier , Beilstein J. Org. Chem., Volume 8, p.421–427, No. 47, (2012)

Synthesis of Mannosylated Glycodendrimers and Evaluation against BC2L-A Lectin from Burkholderia Cenocepacia., Pifferi, Carlo, Goyard David, Gillon Emilie, Imberty Anne, and Renaudet Olivier , Chempluschem, Volume 82, Number 3, p.390–398, (2017)

Synthesis of multi-antigenic platforms as vaccine candidates against cancers., Fiore, Michele, Thomas Baptiste, Dulery Vincent, Dumy Pascal, and Renaudet Olivier , New J. Chem., Volume 37, Number 2, p.286–289, (2013)

Synthesis of Multivalent Glycoconjugates Containing the Immunoactive LELTE Peptide: Effect of Glycosylation on Cellular Activation and Natural Killing by Human Peripheral Blood Mononuclear Cells., Renaudet, Olivier, Krenek Karel, Bossu Isabelle, Dumy Pascal, Kadek Alan, Adamek David, Vanek Ondrej, Kavan Daniel, Gazak Radek, Sulc Miroslav, et al. , J. Am. Chem. Soc., Volume 132, Number 19, p.6800–6808, (2010)

Synthesis of Multivalent Glycoconjugates Containing the Immunoactive LELTE Peptide: Effect of Glycosylation on Cellular Activation and Natural Killing by Human Peripheral Blood Mononuclear Cells [Retraction of document cited in CA152:592290]., Renaudet, Olivier, Krenek Karel, Bossu Isabelle, Dumy Pascal, Kadek Alan, Adamek David, Vanek Ondrej, Kavan Daniel, Gazak Radek, Sulc Miroslav, et al. , J. Am. Chem. Soc., Volume 136, Number 3, p.1156, (2014)

Tailor-made Janus lectin with dual avidity assembles glycoconjugate multilayers and crosslinks protocells., Ribeiro, Joao P., Villringer Sarah, Goyard David, Guerente Liliane, Hoferlin Manuela, Renaudet Olivier, Romer Winfried, and Imberty Anne. , Chem. Sci., Volume 9, Number 39, p.7634–7641, (2018)

Targeting Tn-Antigen-Positive Human Tumors with a Recombinant Human Macrophage Galactose C-Type Lectin, Bulteau, François, Thepaut Michel, Henry Maxime, Hurbin Amandine, Vanwonterghem Laetitia, Vivès Corinne, Le Roy Aline, Ebel Christine, Renaudet Olivier, Fieschi Franck, et al. , Molecular Pharmaceutics, Volume 19, p.235-245, (2022)

Tetravalent glycocyclopeptide with nanomolar affinity to wheat germ agglutinin., Fiore, Michele, Berthet Nathalie, Marra Alberto, Gillon Emilie, Dumy Pascal, Dondoni Alessandro, Imberty Anne, and Renaudet Olivier , Org. Biomol. Chem., Volume 11, Number 41, p.7113–7122, (2013)

Thiol-ene and thiol-yne-based synthesis of glycodendrimers as nanomolar inhibitors of wheat germ agglutinin., Ghirardello, Mattia, Oeberg Kim, Staderini Samuele, Renaudet Olivier, Berthet Nathalie, Dumy Pascal, Hed Yvonne, Marra Alberto, Malkoch Michael, and Dondoni Alessandro. , J. Polym. Sci. Part A Polym. Chem., Volume 52, Number 17, p.2422–2433, (2014)

Thiyl Glycosylation of Propargylated Octasilsesquioxane: Synthesis and Lectin-Binding Properties of Densely Glycosylated Clusters on a Cubic Platform., Marra, Alberto, Staderini Samuele, Berthet Nathalie, Dumy Pascal, Renaudet Olivier, and Dondoni Alessandro. , European J. Org. Chem., Volume 2013, Number 6, p.1144–1149, (2013)

Towards the preparation of synthetic outer membrane vesicle models with micromolar affinity to wheat germ agglutinin using a dialkyl thioglycoside, Fayolle, Dimitri, Berthet Nathalie, Doumeche Bastien, Renaudet Olivier, Strazewski Peter, and Fiore Michele , Beilstein Journal of Organic Chemistry, Volume 15, p.937-946, (2019)

Towards the preparation of synthetic outer membrane vesicle models with micromolar affinity to wheat germ agglutinin using a dialkyl thioglycoside., Fayolle, Dimitri, Berthet Nathalie, Doumeche Bastien, Renaudet Olivier, Strazewski Peter, and Fiore Michele. , Beilstein J. Org. Chem., Volume 15, p.937–946, (2019)

X-Ray Structure of the Key Synthetic Intermediate of a Cancer-Related Sialyl-Tn Antigen Analogue., Renaudet, Olivier, Philouze Christian, Bailly Corinne, Durif Andre, and Dumy Pascal , J. Chem. Crystallogr., Volume 41, Number 2, p.204–208, (2011)